Bioactivity | μ/κ/δ opioid receptor agonist 1 is a μ opioid receptor (MOR), κ opioid receptor (KOR), and δ opioid receptor (DOR) agonist. μ/κ/δ opioid receptor agonist 1 produces a strong and long-lasting analgesic effect through peripheral MOR and KOR in the tail-flick test[1]. |
Name | μ/κ/δ opioid receptor agonist 1 |
Sequence | Tyr-cyclo({d-Lys}-Gly-{p-F-Phe}-Asp)-{d-Pro}-NH2 |
Shortening | Y-cyclo({d-Lys}-G-{p-F-Phe}-D)-{d-Pro}-NH2 |
Formula | C35H45FN8O8 |
Molar Mass | 724.78 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Zhang Q, et al. Structure-Activity Relationships of a Novel Cyclic Hexapeptide That Exhibits Multifunctional Opioid Agonism and Produces Potent Antinociceptive Activity. J Med Chem. 2024 Jan 11;67(1):272-288. |