Bioactivity | Tankyrase-IN-3 is a tankyrase 1 (TNKS1) inhibitor with an IC50 value of 22 nM. Tankyrase-IN-3 can be used for the research of cancer[1]. |
Invitro | Tankyrase-IN-3 具有 TNKS1 抑制活性,IC50 值为 22 nM[1]。 |
Name | Tankyrase-IN-3 |
CAS | 938893-79-9 |
Formula | C21H21N5O4 |
Molar Mass | 407.42 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Alba L Montoya, et al. Combining pharmacophore models derived from DNA-encoded chemical libraries with structure-based exploration to predict Tankyrase 1 inhibitors. Eur J Med Chem. 2023 Jan 15;246:114980. |