Bioactivity | Tankyrase-IN-4 is a tankyrase 1 (TNKS1) inhibitor with an IC50 value of 0.8 nM. Tankyrase-IN-4 can be used for the research of cancer[1]. |
Invitro | Tankyrase-IN-4 具有 TNKS1 抑制活性,IC50 值为 0.8 nM[1]。 |
Name | Tankyrase-IN-4 |
Formula | C25H24N6O5 |
Molar Mass | 488.50 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Alba L Montoya, et al. Combining pharmacophore models derived from DNA-encoded chemical libraries with structure-based exploration to predict Tankyrase 1 inhibitors. Eur J Med Chem. 2023 Jan 15;246:114980. |