| Bioactivity | Lobelanidine is an antagonist for nicotinic acetylcholine receptor (nAChR), which inhibits α7 nAChR response and α3β2/α3β4 nAChR responses, with IC50 of 2.8 and 8.2 μM[1]. |
| Target | IC50: 2.8 μM (α7 nAChR), 8.2 μM (α3β2/α3β4 nAChR) |
| CAS | 552-72-7 |
| Formula | C22H29NO2 |
| Molar Mass | 339.47 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Paz C, et al., (-)-Pentylsedinine, a new alkaloid from the leaves of Lobelia tupa with agonist activity at nicotinic acetylcholine receptor[J]. Natural Product Communications, 2015, 10(8): 1934578X1501000810. |
Lobelanidine
CAS: 552-72-7 F: C22H29NO2 W: 339.47
Lobelanidine is an antagonist for nicotinic acetylcholine receptor (nAChR), which inhibits α7 nAChR response and α3β2
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This product is for research use only, not for human use. We do not sell to patients.