| Bioactivity | Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor with an IC50 of 0.5 μM. | ||||||||||||
| Target | IC50: 0.5 μM (Glutaminyl cyclase) | ||||||||||||
| Invitro | Glutaminyl Cyclase Inhibitor 1 is compound 23[1]. | ||||||||||||
| Name | Glutaminyl Cyclase Inhibitor 1 | ||||||||||||
| CAS | 2110449-60-8 | ||||||||||||
| Formula | C21H24FN3O2 | ||||||||||||
| Molar Mass | 369.43 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Li M, et al. Synthesis and Evaluation of Diphenyl Conjugated Imidazole Derivatives as Potential Glutaminyl Cyclase Inhibitors for Treatment of Alzheimer's Disease. J Med Chem. 2017 Aug 10;60(15):6664-6677. |