| Bioactivity | GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1)[1]. |
| Target | Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1). |
| Name | GPR40/FFAR1 modulator 1 |
| CAS | 874755-26-7 |
| Formula | C21H19N5O3 |
| Molar Mass | 389.41 |
| Appearance | Solid |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | 4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
| Reference | [1]. Lückmann M, et al. Molecular dynamics-guided discovery of an ago-allosteric modulator for GPR40/FFAR1. Proc Natl Acad Sci U S A. 2019 Apr 2;116(14):7123-7128. |