Bioactivity | ASPER-29 is Asperphenamate HY-129578 analog. ASPER-29 also is a dual cathepsin L and S inhibitor with IC50 value of 6.03 μM and 5.02 μM, respectively. ASPER-29 can be used for the research of the migration and invasion of cancer[1]. |
Invitro | ASPER-29 具有双重 Cat L 和 S 抑制效力,IC50 值分别为 6.03 μM 和 5.02 μM[1]。ASPER-29 对胰腺癌 BxPC-3 和 PANC-1 细胞显示出明确的抗转移作用[1]。 |
Name | ASPER-29 |
CAS | 2630388-03-1 |
Formula | C31H29BrN2O5S |
Molar Mass | 621.54 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Haoqiang Huang, et al. Design and synthesis of dual cathepsin L and S inhibitors and antimetastatic activity evaluation in pancreatic cancer cells. Bioorg Med Chem Lett. 2022 Nov 23;80:129087. |