| Bioactivity | 5-HT2A receptor agonist-3 is the most selective agonist for the human 5-HT2A receptor yet discovered, with a Ki of 2.5 nM, and with 124-fold selectivity for 5-HT2A over the structurally similar 5-HT2C receptor[1]. |
| Target | 2.5 nM (human 5-HT2A) |
| Name | 5-HT2A receptor agonist-3 |
| CAS | 1391499-52-7 |
| Formula | C21H26BrNO3 |
| Molar Mass | 420.34 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Juncosa JI Jr, et al. Extensive rigid analogue design maps the binding conformation of potent N-benzylphenethylamine 5-HT2A serotonin receptor agonist ligands. ACS Chem Neurosci. 2013;4(1):96-109. |
5-HT2A receptor agonist-3
CAS: 1391499-52-7 F: C21H26BrNO3 W: 420.34
5-HT2A receptor agonist-3 is the most selective agonist for the human 5-HT2A receptor yet discovered, with a Ki of 2.5 n
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