Bioactivity | β-Chlornaltrexamine dihydrochloride (β-CNA dihydrochloride) is a potent long-term opioid receptor blocker. β-Chlornaltrexamine dihydrochloride can effectively block the inhibitory effect of κ opioid receptor agonists on dopamine release. β-Chlornaltrexamine dihydrochloride can be used to study the mechanism of pain perception[1]. |
CAS | 67025-98-3 |
Formula | C24H34Cl4N2O3 |
Molar Mass | 540.35 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Reichard K L, et al. Regulation of kappa opioid receptor inactivation depends on sex and cellular site of antagonist action[J]. Molecular Pharmacology, 2020, 98(5): 548-558. |