| Bioactivity | mGAT3/4-IN-2 (compound 27b) is a potent mGAT3/mGAT4 inhibitor, with pIC50 values of 5.44 and 5.25, respectively[1]. |
| Target | pIC50: 5.12 ± 0.08 (mGAT1), 5.14 ± 0.07 (mGAT2), 5.44 ± 0.08 (mGAT3), 5.25 ± 0.04 (mGAT4) |
| Name | mGAT3/4-IN-2 |
| CAS | 2556833-68-0 |
| Formula | C26H32ClN3OS2 |
| Molar Mass | 502.13 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Zaręba P, et al. Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice. Eur J Med Chem. 2020 Feb 15;188:111920. |