| Bioactivity | Vasopressin V2 receptor antagonist 2 (Compound 33) is an antagonist of the arginine vasopressin V2 receptor (V2R) with a Ki value of 6.2 nM. Vasopressin V2 receptor antagonist 2 can effectively reduce cAMP levels, thereby inhibiting the growth of renal cysts[1]. |
| Target | Ki: 6.2 nM (V2 receptor). |
| Formula | C62H91FN16O11 |
| Molar Mass | 1255.48 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Xiong X, et al. Long-Residence Time Peptide Antagonist for the Vasopressin V2 Receptor to Treat Autosomal Dominant Polycystic Kidney Disease. J Med Chem. 2024;67(7):5935-5944. |
Vasopressin V2 receptor antagonist 2
CAS: F: C62H91FN16O11 W: 1255.48
Vasopressin V2 receptor antagonist 2 (Compound 33) is an antagonist of the arginine vasopressin V2 receptor (V2R) with a
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