| Bioactivity | VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM. VU 0255035 reduces pilocarpine-induced seizures in mice. VU0255035 is used to examine the role of the M1 receptor in diverse situations[1]. |
| Name | VU 0255035 |
| CAS | 1135243-19-4 |
| Formula | C18H20N6O3S2 |
| Molar Mass | 432.52 |
| Appearance | Solid |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | 4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
| Reference | [1]. Sheffler DJ, et al. A novel selective muscarinic acetylcholine receptor subtype 1 antagonist reduces seizures without impairing hippocampus-dependent learning. Mol Pharmacol. 2009 Aug;76(2):356-68. |
VU 0255035
CAS: 1135243-19-4 F: C18H20N6O3S2 W: 432.52
VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130
Data collection：peptidedb@qq.com
This product is for research use only, not for human use. We do not sell to patients.