| Bioactivity | TCS JNK 5a is a potent JNK3 inhibitor with a pIC50 of 6.7. TCS JNK 5a also inhibits JNK2 with a pIC50 of 6.5. | ||||||||||||
| Invitro | TCS JNK 5a is also screened in a panel of more than 30 kinase assays, including Alk5, c-Fms, CDK-2, EGFR, ErbB2, GSK3β, PLK1, Src, Tie-2 and VegFr2, and is inactive (pIC50<5.0) against all of them[1]. | ||||||||||||
| Name | TCS JNK 5a | ||||||||||||
| CAS | 312917-14-9 | ||||||||||||
| Formula | C20H16N2OS | ||||||||||||
| Molar Mass | 332.42 | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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