Bioactivity | TASP0412098 is an orally available, potent and selective CRTH2/DP2 antagonist with high binding affinity (IC50 2.1 nM) and functional activity (IC50 12 nM). TASP0412098 has the potential to suppress asthma in mouse and guinea pig bronchial asthma models[1]. |
Target | CRTH2/DP2 |
CAS | 1233248-29-7 |
Formula | C27H23ClN2O3 |
Molar Mass | 458.94 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |