Bioactivity | S07-2009 is a potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitor with an IC50 value of 0.20 μM[1]. |
Target | IC50: 0.20 ± 0.12 μM (AKR1C3), 11.18 ± 4.39 μM (AKR1C1), 5.71 ± 2.78 μM (AKR1C2) |
Name | S07-2009 |
CAS | 1580241-55-9 |
Formula | C16H19N3O5 |
Molar Mass | 333.34 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Siyu He, et al. Discovery of Novel Aldo-Keto Reductase 1C3 Inhibitors as Chemotherapeutic Potentiators for Cancer Drug Resistance. ACS Med. Chem. Lett. Jun 2022. |