| Bioactivity | RXFP1 receptor agonist-8 (Example 2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-8 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1.8 nM[1]. |
| Name | RXFP1 receptor agonist-8 |
| CAS | 2941271-76-5 |
| Formula | C40H36F5N3O7 |
| Molar Mass | 765.72 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Jones, Clifford D., et al. Prepration of pyridopyrimidines as KRAS mutant proteins inhibitors useful in treatment of cancers. Patent. WO2022248885. |