| Bioactivity | R8605 is an inhibitor for PKC with an IC50 of 65 μM for PKC in rat brain. R8605 inhibits calcium/phospholipid-independent phosphorylation of protamine with IC50 of 70 μM and 100 μM. R8605 can be used in cancer research[1]. |
| CAS | 119306-51-3 |
| Formula | C22H27NO4 |
| Molar Mass | 369.45 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Sun S. The inhibitory effect of a third generation retinoid, R8605, on protein kinase C activity in vitro[J]. Zhongguo yi xue ke xue Yuan xue bao. Acta Academiae Medicinae Sinicae, 1991, 13(4): 267-270. |