Bioactivity | Pipazethate (SKF 70230A; SQ 15874) hydrochloride is a potent GABA antagonist. Pipazethate hydrochloride shows antitussive activity and can be used in research in cough suppressant [1][2]. |
CAS | 6056-11-7 |
Formula | C21H26ClN3O3S |
Molar Mass | 435.97 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Squires RF, et al. Antidepressants and metabolites that block GABAA receptors coupled to 35S-t-butylbicyclophosphorothionate binding sites in rat brain. Brain Res. 1988 Feb 16;441(1-2):15-22. doi: 10.1016/0006-8993(88)91378-9. [2]. Vakil BJ, et al. Trial of pipazethate as an antitussive. Clin Pharmacol Ther. 1966 Jul-Aug;7(4):515-9. |