Bioactivity | PSB11 hydrochloride is an antagonist with reverse excitatory activity for human A3 Adenosine Receptor with high affinity (Ki=2.3 nM)[1]. |
Name | PSB11 hydrochloride |
CAS | 453591-58-7 |
Formula | C16H18ClN5O |
Molar Mass | 331.80 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Müller C E, et al. [3H] 8-Ethyl-4-methyl-2-phenyl-(8R)-4, 5, 7, 8-tetrahydro-1H-imidazo [2, 1-i]-purin-5-one ([3H] PSB-11), a novel high-affinity antagonist radioligand for human A3 adenosine receptors[J]. Bioorganic & medicinal chemistry letters, 2002, 12(3): 501-503. |