| Bioactivity | PSA-IN-1 (compound 19) is a puromycin sensitive aminopeptidase (PSA) inhibitor with IC50 at 7 nM. PSA-IN-1 has analgesic activity[1]. |
| In Vivo | PSA-IN-1 (50 or 100 μg/mouse, 脑室给药) 单独或与 Met -脑啡肽联用可显著降低小鼠疼痛反应[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
| Formula | C28H32ClN7O3S |
| Molar Mass | 582.12 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Singh R, et al. Modulation of endogenous opioid signaling by inhibitors of puromycin sensitive aminopeptidase. bioRxiv [Preprint]. 2024 Apr 3:2024.04.02.587756. |