Bioactivity | PROTAC FLT-3 degrader 1 is a von Hippel-Lindau-based PROTAC FLT-3 internal tandem duplication (ITD) degrader with an IC50 0.6 nM. Anti-proliferative activity; apoptosis induction[1]. | ||||||||||||
Name | PROTAC FLT-3 degrader 1 | ||||||||||||
CAS | 2230826-81-8 | ||||||||||||
Formula | C52H61N9O9S2 | ||||||||||||
Molar Mass | 1020.23 | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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