| Bioactivity | PROTAC BRM/BRG1 degrader-4 (example 047) is a potent BRM and BRG1 PROTAC degrader, with DC50 values of 0.21 nM and 3.4 nM in SW1573 cells, respectively (Pink: ligand for target protein (HY-168252); Black: linker (HY-28911); Blue: E3 ligase ligand (HY-168253))[1]. |
| Formula | C44H52N10O6S |
| Molar Mass | 849.01 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Peng Gu, et al. Brm selective degradation agent compound and use thereof. WO2023093728A1. |
PROTAC BRM/BRG1 degrader-4
CAS: F: C44H52N10O6S W: 849.01
PROTAC BRM/BRG1 degrader-4 (example 047) is a potent BRM and BRG1 PROTAC degrader, with DC50 values of 0.21 nM and 3.4 n
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