| Bioactivity | PI5P4Ks-IN-3 (compound 30) is a covalent inhibitor of PI5P4K with IC50s of 1.34 μM (PI5P4Kα)，and 9.9 μM (PI5P4Kβ)，respectively. PI5P4Ks-IN-3 shows weak cellular activity[1]. |
| Target | IC50: 1.34 μM (PI5P4Kα), and 9.9 μM (PI5P4Kβ) |
| Name | PI5P4Ks-IN-3 |
| CAS | 2471969-07-8 |
| Formula | C32H31N7O2 |
| Molar Mass | 545.63 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Manz TD, et al. Structure-Activity Relationship Study of Covalent Pan-phosphatidylinositol 5-Phosphate 4-Kinase Inhibitors. ACS Med Chem Lett. 2019 Nov 3;11(3):346-352. |