| Bioactivity | PCSK9-IN-12 is a heteroaryl compound. PCSK9-IN-12 has bind affinity for PCSK9 with a Kd value of <200 nM. PCSK9-IN-12 can be used for the research of cholesterol metabolism[1]. | |||||||||
| Invitro | PCSK9-IN-12 (compound 458B) 对 PCSK9 具有亲和力,Kd 值为 <200 nM[1]。 | |||||||||
| Name | PCSK9-IN-12 | |||||||||
| CAS | 2455427-91-3 | |||||||||
| Formula | C20H20F2N6O2 | |||||||||
| Molar Mass | 414.41 | |||||||||
| Appearance | Solid | |||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | |||||||||
| Storage |
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| Reference | [1]. Michael H. Serrano-Wu, et al. Pcsk9 inhibitors and methods of use thereof. Patent. WO2020150474A1. |