| Bioactivity | P2X7 receptor antagonist-3 is a potent P2X7 receptor antagonist with P2X7R IC50 values of 4.2 nM in humans and 6.8 nM in rats[1]. |
| Name | P2X7 receptor antagonist-3 |
| CAS | 1627900-92-8 |
| Formula | C17H12ClF3N6O |
| Molar Mass | 408.76 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Brad M Savall, et al. Synthesis, SAR, and Pharmacological Characterization of Brain Penetrant P2X7 Receptor Antagonists. ACS Med Chem Lett. 2015 Apr 24;6(6):671-6. |
P2X7 receptor antagonist-3
CAS: 1627900-92-8 F: C17H12ClF3N6O W: 408.76
P2X7 receptor antagonist-3 is a potent P2X7 receptor antagonist with P2X7R IC50 values of 4.2 nM in humans and 6.8 nM in
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