| Bioactivity | Orexin receptor antagonist 4 is potent and selective orexin 2 receptor (OX2R) antagonist with an IC50 of 4.27 nM. Orexin receptor antagonist 4 is 61-fold selective for the OX2R over the OX1R (IC50 of 295 nM) (WO2018206959A1; example 1)[1]. |
| Name | Orexin receptor antagonist 4 |
| CAS | 2251017-69-1 |
| Formula | C23H25FN4O2 |
| Molar Mass | 408.47 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. David Sheppard, et al. Orexin receptor antagonists. WO2018206959A1 |
Orexin receptor antagonist 4
CAS: 2251017-69-1 F: C23H25FN4O2 W: 408.47
Orexin receptor antagonist 4 ispotent and selective orexin 2 receptor (OX2R) antagonist with an IC50 of 4.27 nM. Orexin
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