| Bioactivity | Opioid receptor antagonist 1 (Compound 10) is an Orvinol (HY-D0168)-based opioid receptor antagonist. Opioid receptor antagonist 1 has antagonistic activity to the analgesic properties of Morphine[1]. |
| In Vivo | Opioid receptor antagonist 1 (0.1-10 mg/kg，皮下注射) 剂量依赖性地抑制吗啡对小鼠的镇痛作用 (尾部触击测试)[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
| CAS | 1559075-15-8 |
| Formula | C24H29ClF3NO4 |
| Molar Mass | 487.94 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Ambartsumyan AA, et al. Orvinol-based opioid receptor antagonist fluorinated at C(20)-pharmacophore. Eur J Med Chem. 2024 Dec 18;284:117189. |
Opioid receptor antagonist 1
CAS: 1559075-15-8 F: C24H29ClF3NO4 W: 487.94
Opioid receptor antagonist 1 (Compound 10) is an Orvinol (HY-D0168)-based opioid receptor antagonist. Opioid receptor an
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