| Bioactivity | NPFF2-R ligand 1 (Compound 16a) is a NPFF2-R ligand, with Kis of 228 and 27 nM for NPFF1-R and NPFF2-R respectively. NPFF2-R ligand 1 can be used for research related with central nervous system[1]. |
| Invitro | NPFF2-R ligand 1 对 DOR, KOR and MOR 的结合活性较弱，Ki 值分别为 >10000, 913, 2180 nM[1]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. 0 --> NPFF2-R ligand 1 相关抗体: |
| Formula | C32H41N3O |
| Molar Mass | 483.69 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Galal KA, et al. Guanidine-to-piperidine switch affords high affinity small molecule NPFF ligands with preference for NPFF1-R and NPFF2-R subtypes. Eur J Med Chem. 2024 Mar 23;269:116330. |