Bioactivity | NCRW0005-F05 is a potent GPR139 antagonist with an IC50 value of 0.21 μM. NCRW0005-F05 can be used to research diabetes, obesity and Parkinson's disease[1]. | |||||||||
Target | IC50: 0.21 μM (GPR139) | |||||||||
Name | NCRW0005-F05 | |||||||||
CAS | 342779-66-2 | |||||||||
Formula | C16H13F2NO2 | |||||||||
Molar Mass | 289.28 | |||||||||
Appearance | Solid | |||||||||
Transport | Room temperature in continental US; may vary elsewhere. | |||||||||
Storage |
|
|||||||||
Reference | [1]. Wang J, et al. High-throughput screening of antagonists for the orphan G-protein coupled receptor GPR139. Acta Pharmacol Sin. 2015 Jul;36(7):874-8. |