Bioactivity | N6-Ethyladenosine is an adenosine derivative, acts as a Adenosine receptor agonist, with Kis of 4.9 and 4.7 nM for hA1AR and hA3AR, respectively[1]. | ||||||||||||
Target | Ki: 4.9 nM (hA1AR), 4.7 nM (hA3AR) | ||||||||||||
Invitro | N6-Ethyladenosine (Compound 28) exhibits more selectivity at hA1AR and hA3AR over hA2AR (Ki, 8900±770 nM)[1]. | ||||||||||||
Name | N6-Ethyladenosine | ||||||||||||
CAS | 14357-08-5 | ||||||||||||
Formula | C12H17N5O4 | ||||||||||||
Molar Mass | 295.29 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Kimand SK, et al. Three-dimensional quantitative structure-activity relationship of nucleosides acting at the A3 adenosine receptor: analysis of binding and relative efficacy. J Chem Inf Model. 2007 May-Jun;47(3):1225-33. Epub 2007 Mar 6. |