Bioactivity | Me-(S,R,S)-AHPC-CO-CH2-Br is an E3 ligase ligand-linker conjugate. Me-(S,R,S)-AHPC-CO-CH2-Br can be used to synthesize JNJ-1013 (HY-153188)[1]. |
Formula | C25H33BrN4O4S |
Molar Mass | 565.52 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Fu L, et al. Discovery of highly potent and selective IRAK1 degraders to probe scaffolding functions of IRAK1 in ABC DLBCL[J]. Journal of Medicinal Chemistry, 2021, 64(15): 10878-10889. |