| Bioactivity | MOR agonist-1 is a MOR (μ-opioid receptor) agonist. MOR agonist-1 has good analgesic effect. MOR agonist-1 can be used for the research of pain and pain-related disorders[1]. |
| Invitro | MOR agonist-1 对人类 μ 亚型阿片受体 (hMOR) 具有 cAMP 激动剂活性，EC50 值为 o.5 nM[1]。MOR agonist-1 对 CYP2C19、CYP2D6 和 CYP3A4 具有抑制活性，IC50 值分别为 33.7 μM、12.7 μM 和 40.6 μM[1]。 |
| In Vivo | MOR agonist-1 has good pharmacokinetic properties in rats[1]. |
| Name | MOR agonist-1 |
| CAS | 2305781-14-8 |
| Formula | C22H26ClFN2O2 |
| Molar Mass | 404.91 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. 张杨等，2 ,6-二氧杂螺[4 ,5]癸烷类衍生物、其制备方法及其在医药上的应用。专利，CN115093428A。 |
MOR agonist-1
CAS: 2305781-14-8 F: C22H26ClFN2O2 W: 404.91
MOR agonist-1 is a MOR (μ-opioid receptor) agonist. MOR agonist-1 has good analgesic effect. MOR agonist-1 can be used
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