| Bioactivity | MMP-1-IN-1 (Compound 6) is a highly potent MMP-1 inhibitor with an IC50 of 0.034 μM[1]. |
| Invitro | MMP-1-IN-1 (Compound 6) 对 MMP-1 的高抑制活性可能是由于 MMP-1-IN-1 的 Cl 取代基与 MMP-1 残基 ARG214 之间的卤素键相互作用[1]。 |
| Name | MMP-1-IN-1 |
| Formula | C14H17ClN2O3 |
| Molar Mass | 296.75 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Umedera K, et al. Design of MMP-1 inhibitors via SAR transfer and experimental validation. Sci Rep. 2022 Dec 3;12(1):20915. |