| Bioactivity | MEN 10207 is a selective NK-2 tachykinin receptor (Neurokinin Receptor)?antagonist. MEN 10207 has pA2 values of 5.2, 7.9 and 4.9 in three monoreceptor in vitro assays for NK-1, NK-2 and NK-3 tachykinin receptors, respectively[1][2]. |
| Invitro | In competitive radioligand binding assays, MEN 10207 (the IC50 ranges of 21-54 nM) has high affinity in bovine stomach membranes and SKLKB82#3 cells, a murine fibroblast cell line transfected with a cDNA encoding for the bovine NK2 receptor[3]. |
| Name | MEN 10207 |
| CAS | 126050-12-2 |
| Formula | C57H68N14O10 |
| Molar Mass | 1109.24 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
MEN 10207
CAS: 126050-12-2 F: C57H68N14O10 W: 1109.24
MEN 10207 is a selective NK-2 tachykinin receptor (Neurokinin Receptor)?antagonist. MEN 10207 has pA2 values of 5.2, 7.9
Sales Email：peptidedb@qq.com
This product is for research use only, not for human use. We do not sell to patients.