| Bioactivity | Loperamide (ADL 2-1294) is a selective μ opioid receptor agonist with Kis of 3, 48 and 1156 nM against μ, δ and κ opioid receptor, respectively. Loperamide can be used as an antidiarrheal agent[1]. |
| Target | Ki: 3 nM (μ opioid receptor), 48 nM (δ opioid receptor), 1156 nM (κ opioid receptor) |
| Name | Loperamide |
| CAS | 53179-11-6 |
| Formula | C29H33ClN2O2 |
| Molar Mass | 477.04 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. DeHaven-Hudkins DL, et al. Loperamide (ADL 2-1294), an opioid antihyperalgesic agent with peripheral selectivity. J Pharmacol Exp Ther. 1999 Apr;289(1):494-502. |
Loperamide
CAS: 53179-11-6 F: C29H33ClN2O2 W: 477.04
Loperamide (ADL 2-1294) is a selective μ opioid receptor agonist withKis of 3, 48 and 1156 nM against μ, δ and κ opi
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