| Bioactivity | LP-403812 is a high affinity proline transporter (PROT) inhibitor that produces dose-dependent inhibition of hPROT (IC50=0.11 μM; Ki=0.12 μM) and also inhibits the activity of mouse brain synaptosomal mPROT with the same potency (IC50=0.23 μM). LP-403812 can be used to study the function of PROT in the brain[1]. |
| Target | IC50: 0.11 µM (hPROT) |
| CAS | 1142050-84-7 |
| Formula | C26H34N6O2S |
| Molar Mass | 494.65 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. XuanChuan Yu, et al. "Discovery and characterization of potent small molecule inhibitors of the high affinity proline transporter." Neuroscience letters 451.3 (2009): 212-216. |
LP-403812
CAS: 1142050-84-7 F: C26H34N6O2S W: 494.65
LP-403812 is a high affinity proline transporter (PROT) inhibitor that produces dose-dependent inhibition of hPROT (IC50
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