| Bioactivity | LAU159 is a functionally selective positive modulator of α1β3 GABA(A) receptor with an EC50 of 2.2 μM[1]. |
| Target | EC50: 2.2 μM (α1β3 GABA(A) receptor) |
| Name | LAU159 |
| CAS | 2055050-87-6 |
| Formula | C17H12ClN3O2 |
| Molar Mass | 325.75 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Varagic Z, et al. Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface. Br J Pharmacol. 2013 May;169(2):371-83. |