| Bioactivity | L 888607 Racemate is a selective prostaglandin D2 receptor subtype 1 (DP1) antagonist, with Kis of 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively. | ||||||||||||
| Invitro | L 888607 Racemate (compound 3) maintains a modest binding affinity for the DP1 receptor (Ki = 132 nM) and is actually 8-fold more potent on the TP receptor (Ki = 17 nM)[1]. | ||||||||||||
| Name | L 888607 Racemate | ||||||||||||
| CAS | 1030017-51-6 | ||||||||||||
| Formula | C19H15ClFNO2S | ||||||||||||
| Molar Mass | 375.84 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Beaulieu C, et al. Identification of prostaglandin D2 receptor antagonists based on a tetrahydropyridoindole scaffold. Bioorg Med Chem Lett. 2008 Apr 15;18(8):2696-700. |
L 888607 Racemate
CAS: 1030017-51-6 F: C19H15ClFNO2S W: 375.84
L 888607 Racemate is a selective prostaglandin D2 receptor subtype 1 (DP1) antagonist, with Kis of 132 nM and 17 nM for
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