Bioactivity | HER2-IN-20 (compound 32) is a potent and selective HER2WT and HER2YVMA inhibitor with IC50 values of 49, 42 nM, respectively. HER2-IN-20 has the potential for the research of non-small cell lung cancer (NSCLC)[1]. |
Formula | C30H27ClFN7O2 |
Molar Mass | 572.03 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Hicken EJ, et al. Discovery of Potent and Selective Covalent Inhibitors of HER2WT and HER2YVMA. J Med Chem. 2024 May 31. |