| Bioactivity | Galectin-3 antagonist 1 (compound 15) is a potent and selective Galectin-3 (Gal-3) antagonist with Kd value of 5.3 μM. Meanwhile, Galectin-3 antagonist 1 binds to various Galectin with Kd values of 250 μM (Gal-4N), 18 μM (Gal-4C), 450 μM (Gal-8C), respectively[1]. |
| Target | Kd: 5.3 μM (Gal-3), 250 μM (Gal-4N), 18 μM (Gal-4C), 450 μM (Gal-8C) |
| Name | Galectin-3 antagonist 1 |
| CAS | 2921603-03-2 |
| Formula | C22H22ClNO10 |
| Molar Mass | 495.86 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Bum-Erdene K, et al. Novel Selective Galectin-3 Antagonists Are Cytotoxic to Acute Lymphoblastic Leukemia. J Med Chem. 2022 Apr 28;65(8):5975-5989. |
Galectin-3 antagonist 1
CAS: 2921603-03-2 F: C22H22ClNO10 W: 495.86
Galectin-3 antagonist 1 (compound 15) is a potent and selective Galectin-3 (Gal-3) antagonist with Kd value of 5.3 μM.
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