| Bioactivity | Galantide TFA is a reversible and non-specific galanin (GAL) receptor antagonist. Galantide TFA dose-dependently shows antagonism to galanin-induced K+ conductance with an IC50 value of 4 nM. Galantide TFA can be used for the research of neurological disease and hormone metabolism research[1][2]. | ||||||
| Invitro | Galantide TFA (0.1-10000 nM) 抑制甘丙肽诱导的 K+ 电导的激活,IC50 值为 4 nM[1]。Galantide TFA (0.1-10000 nM) 剂量依赖性地抑制电压依赖性 Ba2+ 电流,IC50 值为 16 nM[1]。Galantide TFA (0.1-10000 nM) 对电压依赖性 Ba2+ 电流的最大抑制率约为 40%[1]。 | ||||||
| Name | Galantide TFA | ||||||
| Formula | C106H152F3N25O28S | ||||||
| Molar Mass | 2313.55 | ||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||
| Storage | Sealed storage, away from moisture and light, under nitrogen
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light, under nitrogen) |