| Bioactivity | GSK3395879 is a selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with an IC50 of 1 nM for hTRPV4[1]. |
| Target | IC50: 1 nM (hTRPV4) |
| Name | GSK3395879 |
| CAS | 2215852-91-6 |
| Formula | C20H15F4N3O5S |
| Molar Mass | 485.41 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Brnardic EJ, et al. Discovery of Pyrrolidine Sulfonamides as Selective and Orally Bioavailable Antagonists of Transient Receptor Potential Vanilloid-4 (TRPV4). J Med Chem. 2018 Nov 8;61(21):9738-9755. |
GSK3395879
CAS: 2215852-91-6 F: C20H15F4N3O5S W: 485.41
GSK3395879 is a selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with an IC
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