| Bioactivity | GSK199 is a reversible and selective PAD4 inhibitor with an IC50 of 200 nM in the absence of calcium[1]. |
| Name | GSK199 |
| CAS | 1549811-53-1 |
| Formula | C24H29ClN6O2 |
| Molar Mass | 468.98 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Lewis HD, et al. Inhibition of PAD4 activity is sufficient to disrupt mouse and human NET formation. Nat Chem Biol. 2015 Mar;11(3):189-91. |