| Bioactivity | GR 64349 is a potent and highly selective NK2 receptor peptide antagonist, with an EC50 of 3.7 nM in rat colon. GR 64349 exhibits selectivity >1000 and >300-fold with respect to NK1 and NK3 receptors, respectively[1][2]. | ||||||
| Name | GR 64349 | ||||||
| CAS | 137593-52-3 | ||||||
| Sequence | Lys-Asp-Ser-Phe-Val-{Aaa}-Leu-Met-NH2 | ||||||
| Shortening | KDSFV{Aaa}LM-NH2 | ||||||
| Formula | C42H68N10O11S | ||||||
| Molar Mass | 921.11 | ||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||
| Storage | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) |