| Bioactivity | GPR35 agonist 1 (compound 50) is a potent and specific G protein-coupled receptor-35 (GPR35)/CXCR8 agonist with an EC50 of 5.8 nM, displays good druggability[1]. |
| Target | EC50: 5.8 nM (GPR35/CXCR8) |
| Name | GPR35 agonist 1 |
| CAS | 2079880-92-3 |
| Formula | C10H4BrN5O5 |
| Molar Mass | 354.07 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Wei L, et al. Discovery of 2H-Chromen-2-one Derivatives as G Protein-Coupled Receptor-35 Agonists. J Med Chem. 2017 Jan 12;60(1):362-372. |