Bioactivity | GPR34 receptor antagonist 2 (Compound D2) is a GPR34 receptor antagonist. GPR34 receptor antagonist 2 can be used for immune diseases, inflammatory diseases research[1]. | ||||||||||||
Target | GPR34 receptor | ||||||||||||
Invitro | Endogenous ligands of GPR34, a G protein-coupled receptor, act on histamine-releasing activity on antigen- or concanavalin A-stimulated rat mast cells and synergize with nerve growth factor on rat mast cells. It is a lipid such as lysophosphatidylserine having the activity of releasing histamine. GPR34 antagonists can be used, for example, for histamine release inhibitors, immune diseases, edema, hyperacidity, etc[1]. | ||||||||||||
Name | GPR34 receptor antagonist 2 | ||||||||||||
CAS | 907952-06-1 | ||||||||||||
Formula | C31H26ClNO4 | ||||||||||||
Molar Mass | 512.00 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Fumio Ito, et al. Agent for controlling function of gpr34 receptor. WO2006088246 A1. |