| Bioactivity | GFB-12811 is a high selective and orally active CDK5 inhibitor with an IC50 of 2.3 nM. GFB-12811 is highly selective over the other tested kinases (CDK1/2/6/7/9)[1]. | ||||||||||||
| Name | GFB-12811 | ||||||||||||
| CAS | 2775311-17-4 | ||||||||||||
| Formula | C22H23F4N5O | ||||||||||||
| Molar Mass | 449.44 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Daniels MH, et al. Discovery and Optimization of Highly Selective Inhibitors of CDK5. J Med Chem. 2022;65(4):3575-3596. |
GFB-12811
CAS: 2775311-17-4 F: C22H23F4N5O W: 449.44
GFB-12811 is a high selective and orally active CDK5 inhibitor with an IC50 of 2.3 nM. GFB-12811 is highly selective ove
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