| Bioactivity | GABAA receptor agent 1 is a high affinity ligand for GABAA receptor, with potent anticonvulsant activity[1]. | ||||||||||||
| In Vivo | GABAA receptor agent 1 (30 mg/kg; intraperitoneal) inhibits the maximum electroshock (MES) and pentylenetetrazole (PTZ)-induced convulsions in swiss albino rats[1]. | ||||||||||||
| Name | GABAA receptor agent 1 | ||||||||||||
| CAS | 1571-87-5 | ||||||||||||
| Formula | C13H8ClN3O2 | ||||||||||||
| Molar Mass | 273.67 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
|
||||||||||||
| Reference | [1]. Jain P, et al. Design, synthesis and biological evaluation of some novel benzimidazole derivatives for their potential anticonvulsant activity. Arch Pharm Res. 2010 Jul;33(7):971-80. |