PeptideDB

Fedovapagon

CAS: 347887-36-9 F: C27H34N4O3 W: 462.58

Fedovapagon (VA106483) is a selective and orally active vasopressin V2 receptor (V2R) agonist with an EC50 of 24 nM. Fed
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This product is for research use only, not for human use. We do not sell to patients.

Bioactivity Fedovapagon (VA106483) is a selective and orally active vasopressin V2 receptor (V2R) agonist with an EC50 of 24 nM. Fedovapagon can be used in the research of nocturia[1].
In Vivo Fedovapagon (1 mg/kg, oral administration) inhibits urine output with 81% inhibition rate in rats[1]. Animal Model:
Name Fedovapagon
CAS 347887-36-9
Formula C27H34N4O3
Molar Mass 462.58
Appearance Solid
Transport Room temperature in continental US; may vary elsewhere.
Storage

4°C, stored under nitrogen

*In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)

Reference [1]. Yea CM, et al. New benzylureas as a novel series of potent, nonpeptidic vasopressin V2 receptor agonists. J Med Chem. 2008 Dec 25;51(24):8124-34.