Bioactivity | ERα degrader 11 (compound B16) is a selective ERα degrader that can be used as an estrogen receptor probe to investigate ER status in ER-positive breast cancer cells[1]. |
CAS | 3052336-87-2 |
Formula | C28H27F3N2O3 |
Molar Mass | 496.52 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Lu Y, et al. Discovery of non-antiproliferative selective estrogen receptor degraders (SERDs) based on scaffold optimization of elacestrant. Eur J Med Chem. 2024 Sep 21;279:116897. |